Access to the nucleus and functional association with c-Myc is required for the full oncogenic potential of ΔEGFR/EGFRvIII

J Biol Chem. 2013 Feb 1;288(5):3428-38. doi: 10.1074/jbc.M112.399352. Epub 2012 Dec 17.

Abstract

ΔEGFR is a potent glioblastoma oncogene which has been studied primarily as a plasma membrane kinase. Using intracranial xenograft studies in mice, we show that blocking ΔEGFR access to the nucleus attenuates its tumorigenicity and, conversely, that promoting nuclear accumulation enhances this, providing the first in vivo evidence that the nuclear actions of ΔEGFR contribute strongly to its oncogenic function. Nuclear actions of ΔEGFR include regulation of gene expression by participation in chromatin-bound complexes, and genome-wide mapping of these sequences by chromatin immunoprecipitation and massively parallel sequencing identified 2294 peaks. Bioinformatic analysis showed enrichment of the E-box motif in the dataset, and c-Myc and ΔEGFR were corecruited to the promoters of and transcriptionally activated a subset of nuclear ΔEGFR chromatin targets. Knockdown of c-Myc decreased the expression of these targets and diminished ΔEGFR-stimulated anchorage-independent colony formation. We conclude that transcriptional regulation of target genes by association with gene regulatory chromatin in cooperation with c-Myc by nuclear ΔEGFR makes a unique contribution to its oncogenicity and propose that this venue provides new targets for therapeutic intervention.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Cell Nucleus / metabolism*
  • Cell Transformation, Neoplastic / metabolism*
  • Cell Transformation, Neoplastic / pathology
  • Chromatin Immunoprecipitation
  • E-Box Elements / genetics
  • ErbB Receptors / chemistry
  • ErbB Receptors / metabolism*
  • Genome, Human / genetics
  • Glioma / metabolism
  • Humans
  • Mice
  • Mice, Nude
  • Mutant Proteins / metabolism
  • Mutation / genetics*
  • Nuclear Export Signals
  • Nuclear Localization Signals / metabolism
  • Phenotype
  • Promoter Regions, Genetic / genetics
  • Protein Binding
  • Protein Multimerization
  • Protein Transport
  • Proto-Oncogene Proteins c-myc / metabolism*
  • Transcription Factors / metabolism

Substances

  • Mutant Proteins
  • Nuclear Export Signals
  • Nuclear Localization Signals
  • Proto-Oncogene Proteins c-myc
  • Transcription Factors
  • epidermal growth factor receptor VIII
  • ErbB Receptors